Amycretin

Investigational GLP-1 / Weight Loss

Novo Nordisk's oral GLP-1/amylin dual agonist showing unprecedented weight loss for an oral medication.

Also Known As
NNC0487-0111
Status
Investigational
Category
GLP-1 / Weight Loss
Route
Oral tablet (investigational)

What Is Amycretin?

Amycretin is an investigational oral peptide developed by Novo Nordisk that combines GLP-1 and amylin receptor agonism in a single molecule. It represents a convergence of two major trends in obesity medicine: dual-receptor targeting (like CagriSema) and oral delivery (like orforglipron).

Amylin is a hormone co-secreted with insulin that promotes satiety, slows gastric emptying, and suppresses glucagon. By combining amylin's mechanisms with GLP-1's powerful appetite suppression and insulin sensitization, amycretin targets multiple metabolic pathways simultaneously. The oral formulation would eliminate the need for injections entirely.

Early clinical data has generated significant excitement: amycretin showed up to 13% weight loss in just 12 weeks in Phase 1 — a rate of weight loss that, if sustained, could rival or exceed injectable agents.

What The Research Says

Phase 1 results presented at conferences showed remarkable weight loss velocity: up to 13% body weight reduction over 12 weeks with oral amycretin. This exceeds the early weight loss trajectory of injectable semaglutide and tirzepatide at comparable time points.

The dual GLP-1/amylin mechanism in oral form is unique. If Phase 2/3 data confirms the Phase 1 trajectory, amycretin could become a game-changing oral obesity treatment. Novo Nordisk has prioritized its development.

Common Uses

Important Safety Information

GI side effects expected (nausea, vomiting). Full safety profile not yet established. Clinical trial use only.

Questions To Ask Your Provider

  1. When are Phase 2 results expected?
  2. How does the weight loss rate compare to injectable agents?
  3. Are clinical trials enrolling?

Regulatory Status

NOT FDA-approved. In Phase 1/2 clinical trials. Novo Nordisk pipeline.

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Disclaimer: This information is for educational purposes only. PepKey does not diagnose, prescribe, or recommend dosages. Always consult a licensed healthcare provider before starting any peptide therapy. Full disclosure
Last updated: 2026-04-08 · ← Back to Peptide Library